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PD-198306
  • 品牌:MedKoo
  • 產(chǎn)地:美國
  • 貨號:525904
  • cas:212631-61-3
  • 發(fā)布日期: 2022-07-20
  • 更新日期: 2024-08-12
產(chǎn)品詳請
產(chǎn)地 美國
品牌 MedKoo
貨號 525904
用途 This product is for research use only, not for human or veterinary use.
包裝規(guī)格 5.0mg;
CAS編號 212631-61-3
純度 >98%%
是否進(jìn)口
CAS No:212631-61-3
分子式:C18H16F3IN2O2
折射率:1.631
密度:1.686
用途:Potent inhibitor of MEK1/2. Inhibits isolated enzyme at a concentration of 8 nM and inhibits MEK activity in synovial fibroblasts at concentrations of 30-100 nM. Highly selective for MEK; IC 50 values are > 1, > 4, > 4 and > 10 μ M for ERK, c-Src, cdks and PI 3-kinase γ respectively. A..