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CBL0137 (CBL-0137)
  • 品牌:MedKoo
  • 產(chǎn)地:美國
  • 貨號:584439
  • cas:1197397-89-9
  • 發(fā)布日期: 2022-07-20
  • 更新日期: 2024-08-12
產(chǎn)品詳請
產(chǎn)地 美國
品牌 MedKoo
貨號 584439
用途 This product is for research use only, not for human or veterinary use.
包裝規(guī)格 5.0mg; 25.0mg;
CAS編號 1197397-89-9
純度 >98%%
是否進(jìn)口
中文名稱:1197397-89-9
CAS No:1197397-89-9
分子式:C21H25ClN2O2
用途:Curaxins are small molecules that simultaneously activate p53 and inhibit NF-κB without causing detectable genotoxicity. CBL0137 is a water soluble and metabolically stable curaxin that activates p53 with an EC50 value of 0.37 μM and inhibits NF-κB with an EC50 value of 0.47 μM. It functionally ..